
Chemical Name : MK8245
CAS : 1030612-90-8
Synonyms: 5-[3-[4-(2-Bromo-5-fluorophenoxy)-1-piperidinyl]-5-isoxazolyl]-2H-tetrazole-2-acetic acid
Solubility:DMSO
Storage:-20°C for 2 years
Biologieal
Stearoyl-CoA desaturase (SCD) inhibitors
Reference
1、Novel, potent, selective, and metabolically stable stearoyl-CoA desaturase (SCD) inhibitors.
By Koltun, Dmitry O.; Parkhill, Eric Q.; et al.
From Bioorganic & Medicinal Chemistry Letters (2009), 19(7), 2048-2052.
2、Discovery of piperidine-aryl urea-based stearoyl-CoA desaturase 1 inhibitors.
By Xin, Zhili; Zhao, Hongyu; et al .
VX-770/VX770
873054-44-5
AZD-7762/AZD7762
860352-01-8
Pimecrolimus/
137071-32-0
Granzyme B Inhibitor Z-AAD-CH2Cl