
化学名称 : MK8245
CAS : 1030612-90-8
英文名称: MK8245
英文同义词: 5-[3-[4-(2-Bromo-5-fluorophenoxy)-1-piperidinyl]-5-isoxazolyl]-2H-tetrazole-2-acetic acid
溶解度:DMSO
储存条件:-20°C for 2 years
生物活性
Stearoyl-CoA desaturase (SCD) inhibitors
参考文献
1、Novel, potent, selective, and metabolically stable stearoyl-CoA desaturase (SCD) inhibitors.
By Koltun, Dmitry O.; Parkhill, Eric Q.; et al.
From Bioorganic & Medicinal Chemistry Letters (2009), 19(7), 2048-2052.
2、Discovery of piperidine-aryl urea-based stearoyl-CoA desaturase 1 inhibitors.
By Xin, Zhili; Zhao, Hongyu; et al .
2-甲氧基-N-[(2E)-3-[4-[[3-甲基-4-[(6-甲基-3-吡啶基)氧基]苯基]氨基]-6-喹唑啉基]-2-丙烯-1-基]乙酰胺
383432-38-0
ARRY-334543/
N-[(4-甲基苯基)磺酰基]-L-精氨酸甲酯
901-47-3
Torin 1
1222998-36-8