
化学名称 : SB408124/SB-408124/
CAS : 288150-92-5
溶解度:Soluble to 100 mM in DMSO
储存条件:Store at RT
生物活性
Selective non-peptide orexin OX1 receptor antagonist (Kb values are 21.7 and 1405 nM for human OX1 and OX2 receptors respectively). Blocks orexin-A induced grooming following oral administration in vivo.
(1S,2R,5R)-5-(4-氨基-1H-咪唑并[4,5-C]吡啶-1-基)-3-羟甲基-3-环戊烯-1,2-二醇
102052-95-9
NNC 756(Odapipam)/
PSNCBAM-1/
GYKI-52466/
102771-26-6