288150-92-5

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SB408124/SB-408124/

288150-92-5

编号ABP000452 化学名称SB408124/SB-408124/ 分子式C19H18F2N4O 分子量356.3692 纯度 >98 %

化学名称 : SB408124/SB-408124/

CAS : 288150-92-5

溶解度:Soluble to 100 mM in DMSO

储存条件:Store at RT

生物活性

Selective non-peptide orexin OX1 receptor antagonist (Kb values are 21.7 and 1405 nM for human OX1 and OX2 receptors respectively). Blocks orexin-A induced grooming following oral administration in vivo.
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