BIX 02188

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BIX 02188

BIX 02188

Cat.No.ABP027337 Chemical NameBIX 02188 CAS334949-59-6 MDL: MFCD14584538 MolFormulaC25H24N4O2 MolWeight412.48 Purity NLT 98%

Chemical Name : BIX 02188

CAS : 334949-59-6

BIX02188 is a selective inhibitor of MEK5 with IC50 of 4.3 nM, also inhibits ERK5 catalytic activity with IC50 of 810 nM, and does not inhibit closely related kinases MEK1, MEK2, ERK2, and JNK2.
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