Selpercatinib

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Selpercatinib

Selpercatinib

编号ABP016514 化学名称Selpercatinib CAS2152628-33-4 分子式 分子量 纯度 NLT 98%

化学名称 : Selpercatinib

CAS : 2152628-33-4

Selpercatinib is a RET kinase inhibitor extracted from patent WO2018071447A1, Compound Example 163, has an IC50 of 14.0 nM, 24.1 nM, and 530.7 nM for RET (WT), RET (V804M) , and RET (G810R), respectively. Antineoplastic activity.
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