
Chemical Name : MK8245
CAS : 1030612-90-8
Synonyms: 5-[3-[4-(2-Bromo-5-fluorophenoxy)-1-piperidinyl]-5-isoxazolyl]-2H-tetrazole-2-acetic acid
Solubility:DMSO
Storage:-20°C for 2 years
Biologieal
Stearoyl-CoA desaturase (SCD) inhibitors
Reference
1、Novel, potent, selective, and metabolically stable stearoyl-CoA desaturase (SCD) inhibitors.
By Koltun, Dmitry O.; Parkhill, Eric Q.; et al.
From Bioorganic & Medicinal Chemistry Letters (2009), 19(7), 2048-2052.
2、Discovery of piperidine-aryl urea-based stearoyl-CoA desaturase 1 inhibitors.
By Xin, Zhili; Zhao, Hongyu; et al .
Triptolide(PG490)/
38748-32-2
Danoprevir(ITMN-191)/RG7227,RO5190591
PNU-282987
123464-89-1
Masitinib/AB1010
790299-79-5