1013101-36-4

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PF-04691502

1013101-36-4

Cat.No.ABP000986 Chemical NamePF-04691502 MDL: MFCD18782794 MolFormulaC22H27N5O4 MolWeight425.486 Purity >99%

Chemical Name : PF-04691502

CAS : 1013101-36-4

Synonyms: 2-Amino-6-(6-methoxypyridin-3-yl)-4-methyl-8-[(1R,4R)-4-(2-hydroxyethoxy)cyclohexyl]-7h,8h-pyrido[2,3-d]pyrimidin-7-one

Solubility:Soluble to 10 mM in DMSO and to 50 mM in ethanol

Storage:Desiccate at +4°C

Biologieal

A selective h5-HT1D antagonist, displaying 60-fold selectivity over h5-HT1B, and exhibiting little or no affinity for a range of other receptor types.

Reference

Hagan et al (1997) Stimulation of 5-HT1B receptors causes hypothermia in the rat. Eur.J.Pharmacol. 331 169. PMID: 9274976.
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