BTRX-335140
编号ABP014525
化学名称BTRX-335140
CAS2244614-14-8
分子式
分子量
纯度 NLT 98%
化学名称 : BTRX-335140
CAS : 2244614-14-8
英文名称: BTRX-335140
英文同义词:
BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. BTRX-335140 endows with favorable in vitro ADMET and in vivo pharmacokinetic profiles and medication-like duration of action in rats.
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