Ocaperidone

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Ocaperidone

Ocaperidone

编号ABP013969 化学名称Ocaperidone CAS129029-23-8 MDL: MFCD00866668 分子式C24H25FN4O2 分子量420.48 纯度 NLT 98%

化学名称 : Ocaperidone

CAS : 129029-23-8

英文名称: Ocaperidone

英文同义词:

Ocaperidone is an effective antipsychotic agent, acting as a potent 5-HT2 and dopamine D2 antagonist, and a 5-HT1A agonist, with Kis of 0.14 nM, 0.46 nM, 0.75 nM, 1.6 nM and 5.4 nM for 5-HT2, a1-adrenergic receptor, dopamine D2, histamine H1 and a2-adrenergic receptor, respectively, and a pEC50 and pKi of 7.60 and 8.08 for h5-HT1A.
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