
化学名称 : Amisulpride/
CAS : 71675-85-9
英文名称: Amisulpride/
英文同义词: 4-Amino-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-(ethylsulfonyl)-2-methoxybenzamide
溶解度:Unknown
储存条件:at -20℃ 2 years
生物活性
Amisulpride is an atypical antipsychotic used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder. In small doses it is also used to treat depression. Amisulpride functions primarily as a D2 and D3 receptor antagonist. It has high affinity for these receptors with dissociation constants of 2.8 nM and 3.2 nM, respectively. [1]
参考文献
[1] http://en.wikipedia.org/wiki/Amisulpride
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