![N-[3-[[5-溴-4-[[2-(1H-咪唑-5-基)乙基]氨基]-2-嘧啶基]氨基]苯基]-1-吡咯烷甲酰胺](https://stcdn.activebiopharma.com/active/ABP000487.png)
化学名称 : N-[3-[[5-溴-4-[[2-(1H-咪唑-5-基)乙基]氨基]-2-嘧啶基]氨基]苯基]-1-吡咯烷甲酰胺
CAS : 702674-56-4
英文名称: BX912/BX-912/
英文同义词: BX-912
生物活性
Inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1).
参考文献
R I Feldman et al. Novel Small Molecule Inhibitors of 3-Phosphoinositide-dependent Kinase-1. J. Biol. Chem., 2005, 280, 20, 19867-19874. C Peifer, D R. Alessi, Small-Molecule Inhibitors of PDK1. ChemMedChem. 2008, 3 (10), Review. [online abstract]
(8R)-8-(3,5-二氟苯基)-10-氧代-N-[(2R)-1,1',2',3-四氢-2'-氧代螺[2H-茚-2,3'-[3H]吡咯并[2,3-b]吡啶]-5-基]-6,9-二氮杂螺[4.5]癸烷-9-乙酰胺盐酸盐
957116-20-0
5-氨基乙酰丙酸
106-60-5
盐酸吉西他滨
122111-03-9
苯磺酸贝托司汀
190786-44-8