化学名称 : BX795
CAS : 702675-74-9
英文名称: BX795/BX-795/
英文同义词: N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide
同义词: N-[3-[[5-碘-4-[[3-[(2-噻吩基羰基)氨基]丙基]氨基]-2-嘧啶基]氨基]苯基]-1-吡咯烷甲酰胺
生物活性
BX 795 was initially developed as a PDK1 inhibitor. Recent study highlighted on its bioactivitiy as a potent and relatively specific inhibitor of TBK1 and closely related IKK
参考文献
R I Feldman et al. Novel Small Molecule Inhibitors of 3-Phosphoinositide-dependent Kinase-1. J. Biol. Chem., 2005, 280, 20, 19867-19874. [online] J Bain et al. The selectivity of protein kinase inhibitors: a further update. Biochem. J. 2007, 408, 297