化学名称 : N-[3-[[5-溴-4-[[2-(1H-咪唑-5-基)乙基]氨基]-2-嘧啶基]氨基]苯基]-1-吡咯烷甲酰胺
CAS : 702674-56-4
英文名称: BX912/BX-912/
英文同义词: BX-912
生物活性
Inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1).
参考文献
R I Feldman et al. Novel Small Molecule Inhibitors of 3-Phosphoinositide-dependent Kinase-1. J. Biol. Chem., 2005, 280, 20, 19867-19874. C Peifer, D R. Alessi, Small-Molecule Inhibitors of PDK1. ChemMedChem. 2008, 3 (10), Review. [online abstract]