
化学名称 : 21-羟基-17-(1-氧代丙氧基)孕甾-4-烯-3,20-二酮
CAS : 19608-29-8
英文名称: 17 alpha-propionate /
英文同义词: 17 ALPHA-PROPIONATE
溶解度:DMSO
储存条件:at -20℃ 2 years
生物活性
Ostarine (MK-2866) is an androgen receptor modulator (SARM) with an ED50 of 0.44 mg/day. Ostarine (MK-2866) has anabolic activity. Lack of PSA increases in men and hair growth in women further corroborated selective anabolic effects of Ostarine (MK-2866). Ostarine (MK-2866) also resulted in a dose-dependent decrease in LDL and HDL cholesterol levels, with the average LDL/HDL ratio for all doses remaining in the low cardiovascular risk catergory. [1][2][3]
参考文献
[1] Zilbermint MF et al. Future Oncol. 2009 Oct; 5(8):1211-20.
[2] Madeddu C et al. Curr Opin Support Palliat Care. 2009 Dec; 3(4):258-62.
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