化学名称 : RJR 2403 oxalate
CAS : 183288-99-5
英文名称: RJR 2403 oxalate
英文同义词: (E)-N-Methyl-4-(3-pyridinyl)-3-bute n-1-amine oxalate
溶解度:Soluble to 100 mM in water
储存条件:Desiccate at +4°C
生物活性
A neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki values are 26 and 36000 nM for α4β2 and α7 receptors respectively). Active in vivo
参考文献
Bencherif et al (1996) RJR-2403: a nicotinic agonist with CNS selectivity I. In vitro characterization. J.Pharmacol.Exp.Ther.