
化学名称 : 西洛多辛
CAS : 160970-54-7
英文名称: Silodosin(Rapaflo)/KAD 3213,KMD 3213
英文同义词: SILODOSIN
溶解度:Unknown
储存条件:at -20℃ 2 years
生物活性
Silodosin(Rapaflo) is an ��1-adrenoceptor antagonist with high uroselectivity. It causes practically no orthostatic hypotension (in contrast to other ��1 blockers). Since Silodosin is a highly selective inhibitor of the ��1A adrenergic receptor, it causes practically no orthostatic hypotension (in contrast to other ��1 blockers). On the other hand, the high selectivity seems to cause more problems with ejaculation. [1]
参考文献
[1] http://en.wikipedia.org/wiki/Silodosin
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