化学名称 : RKI-1447
CAS : 1342278-01-6
英文名称: RKI-1447
英文同义词: 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea
溶解度:Soluble in water and DMSO
储存条件:at -20℃ 2 years
生物活性
Small-molecule antagonist of methyl-lysine (KMe) reader protein with selectivity for L3MBTL1 and L3MBTL3 (IC50 of 4.2μM and 3.1μM respectively, ref 1).