AZ6102

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AZ6102

AZ6102

Cat.No.ABP021073 Chemical NameAZ6102 CAS1645286-75-4 MolFormula MolWeight Purity NLT 98%

Chemical Name : AZ6102

CAS : 1645286-75-4

AZ6102 is a potent dual TNKS1 and TNKS2 inhibitor, with IC50s of 3 nM and 1 nM, respectively, and alao has 100-fold selectivity against other PARP family enzymes, with IC50s of 2.0 μM, 0.5 μM, and >3 μM, for PARP1, PARP2, and PARP6, respectively.
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